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" "A small molecule for theraNOstic targeting of cancer cells " Ravikumar, G.; Bagheri, M.; Saini, D. K.; Chakrapani, H. Chemical Communications 2017, in press, xy-yy

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" "Visible-Light-Triggered Uncaging of Carbonyl Sulfide for Hydrogen Sulfide (H2S) Release" Sharma, A. K.; Nair, M.; Chauhan, P.; Gupta, K.; Saini, D. K.; Chakrapani, H. Organic Letters 2017, 19, 4822-4825

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" "On demand" redox buffering by H2S contributes to antibiotic resistance revealed by a bacteria-specific H2S donor Shukla, P.; Khodade, V. S.; SharathChandra, M.; Chauhan, P.; Mishra, S.; Siddaramappa, S.; Bulagonda, E. P.; Singh, A.; Chakrapani, H. Chemical Science 2017, 8, 4967-4972

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" FLUORO/NO, a Nitric Oxide Donor with a Fluorescence Reporter; Ravikumar, G.; Bagheri, M.; Saini, D. K.; Chakrapani, H. ChemBioChem 2017, 19, 62-65

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" Esterase Activated Carbonyl Sulfide/Hydrogen Sulfide (H2S) Donors; Chauhan, P.; Bora, P.; Ravikumar, G.; Jos, S.; Chakrapani, H. Organic Letters 2017, 19, 62-65

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" A Small Molecule for Controlled Generation of Peroxynitrite; Khodade, V.S.; Kulkarni, A.; Sen Gupta, A.; Sengupta, K.; Chakrapani, H. Organic Letters 2016, 18, 1274-1277

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" Thiol Activated Prodrugs of Sulfur Dioxide (SO2) as MRSA Inhibitors; Pardeshi, K. A.; Malwal, S. R. Banerjee, A.; Lahiri, S.; Rangarajan, R.; Chakrapani, H. Bioorganic and Medicinal Chemistry Letters 2015, 13, 2694-2697

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" Mycobacterium tuberculosis has diminished capacity to counteract redox stress induced by elevated levels of endogenous superoxide; Tyagi, P.; Dharmaraja, A. T.; Bhaskar, A.; Chakrapani, H.; Singh, A. Free Radical Biology and Medicine 2015, 84, 344-354

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" Benzosulfones as Photochemically Activated Sulfur Dioxide (SO2) Donors ; Malwal, S. R. Chakrapani, H. Organic and Biomolecular Chemistry 2015, 13, 2399-2406

Graphical abstract: Benzosulfones as photochemically activated sulfur dioxide (SO2) donors

" A phenacrylate scaffold for tunable thiol activation and release ; Sankar, R. K; Kumbhare, R. S.; Dharmaraja, A. T.; Chakrapani, H. Chemical Communications 2014, 50, 15323-15326

"Substituent Effects on Reactive Oxygen Species (ROS) Generation by Hydroquinones; Dharmaraja, A. T.; Jain, C.; Chakrapani, H. The Journal of Organic Chemistry 2014, 79, 9413-9417

"A Highly Selective Sulfinate Ester Probe for Thiol Bioimaging" Malwal, S. R..; Labade, A.; Andhalkar, A. S.; Sengupta, K.; Chakrapani, H. Chemical Communications 2014, 50, 78, 11533-11535

 “Site-directed delivery of nitric oxide to cancers” Sharma, K.; Chakrapani, H. Nitric Oxide: Biology and Chemistry 2014, xx, in press.

"Bioreductively Activated Reactive Oxygen Species (ROS) Generators as MRSA Inhibitors" Khodade, V. S.; Sharath Chandra, M.; Banerjee, A.; Lahiri, S.; Pulipeta, M.; Rangarajan, R.; Chakrapani, H. ACS Medicinal Chemistry Letters 2014, 5, 777-781

"Arylboronate Ester Based Diazeniumdiolates (BORO/NO), a Class of Hydrogen Peroxide Inducible Nitric Oxide (NO) Donors" Dharmaraja, A. T.; Ravikumar, G.; Chakrapani, H. Organic Letters 2014, 16, 2610-2613

"A Small Molecule for Controlled Generation of Reactive Oxygen Species (ROS)" Dharmaraja, A. T.; Chakrapani, H. Organic Letters 2014, 16, 398-401

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"Nitroreductase-Activated Nitric Oxide Prodrugs" Sharma, K.; Sengupta, K.; Chakrapani, H. Bioorganic and Medicinal Chemistry Letters 2013, 23, 5964-5967

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"INDQ NO, a Bioreductively Activated Nitric Oxide Prodrug" Sharma, K.; Iyer, I.; Sengupta, K.; Chakrapani, H. Organic Letters 2013, 15, 2636-2639

"Benzosultines as Sulfur Dioxide (SO2) Donors" Malwal, S. R.; Gudem, M.; Hazra, A.; Chakrapani, H. Organic Letters 2013, 15, 1116-1119

"Design, Synthesis and Evaluation of Small Molecule Reactive Oxygen Species Generators as Selective Mycobacterium Tuberculosis Inhibitors" Dharmaraja, A. T.; Alvala, M.; Sriram, D.; Yogeeswari, P.; Chakrapani, H. Chemical Communications 48 (2012), pp. 10325-10327

"Synthesis and antimycobacterial activity of prodrugs of sulfur dioxide (SO2)" Malwal, S. R.; Sriram, D.; Yogeeswari, P.; Chakrapani, H. Bioorganic & Medicinal Chemistry Letters 22 (2012), pp. 3603-3606

"Synthesis, reactive oxygen species generation and copper-mediated nuclease activity profiles of 2-aryl-3-amino-1,4-naphthoquinones" Khodade, V. S.; Dharmaraja, A. T.; Chakrapani, H. Bioorganic & Medicinal Chemistry Letters 22 (2012) 3766–3769

"Design, Synthesis and Evaluation of Thiol-Activated Sources of Sulfur Dioxide (SO2) as Antimycobacterial Agents" Malwal, S. R.; Dharmarajan, S.; Yogeeswari, P.; Konkimalla, V. B.;Chakrapani, H. Journal of Medicinal Chemistry 2012, 55, 553-557

"Synthesis, thiol-mediated reactive oxygen species generation profiles and anti-proliferative activities of 2,3-epoxy-1,4-naphthoquinones" Medicinal Chemistry Communications, 2012, 3, 212-216

For complete list of publications, check Publications

 

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